Due to stimulation of the parasympathetic nervous system, bethanechol increases bladder muscle tone causing contractions which initiate urination. Bethanechol also stimulates gastric motility, increases gastric tone and may restore peristalsis.(UTD)
藥動學
禁忌症
asthma
bradycardia, hypotension/vasomotor instability/vagotonia
compromised integrity of gastrointestinal or bladder wall
coronary artery disease
epilepsy
gastrointestinal inflammation, spasms, peritonitis
gastrointestinal or bladder surgery, resection, obstruction
hypersensitivity to bethanechol or components
hyperthyroidism
Parkinsonism
peptic ulcer.
懷孕分類
C (FDA) B2 (AUS)
哺乳分類
Infant risk cannot be ruled out.(MDX)
副作用
Common:
Dermatologic: Flushing
Gastrointestinal: Abdominal cramps, Diarrhea
Renal: Urgent desire to urinate
Serious:
Neurologic: Seizure
Respiratory: Acute exacerbation of asthma
劑量和給藥方法
Urinary retention:
initial, 5 to 10 mg ORALLY repeated hourly until satisfactory response, MAX 50 mg; usual dose range, 10 to 50 mg ORALLY 3 or 4 times daily
initial, 0.5 mL (2.575 mg) SC at 15-30 min intervals until satisfactory response, MAX 4 doses; maintenance, 1 mL (5.15 mg) SC, 3-4 times daily.