局部麻醉 Prevention and control of pain in procedures involving the male and female urethra; for topical treatment of painful urethritis
藥理
Blocks both the initiation and conduction of nerve impulses by decreasing the neuronal membrane's permeability to sodium ions, which results in inhibition of depolarization with resultant blockade of conduction.
藥動學
禁忌症
Sensitivity to local anesthetics of the amide type or to any other component of the product
懷孕分類
B (FDA)
哺乳分類
Compatible with breastfeeding (WHO)
Infant risk is minimal (MDX)
Anesthesia of male urethra: 5 to 30 mL (100 to 600 mg)
Anesthesia of female urethra: 3 to 5 mL (60 to 100 mg)
Maximum dose: 30 mL (600 mg) in any 12-hour period.
小兒調整劑量
Dose varies with age and weight (maximum dose: 4.5 mg/kg)
腎功能調整劑量
There are no dosage adjustments provided in the manufacturer's labeling.
肝功能調整劑量
There are no dosage adjustments provided in the manufacturer's labeling; use caution in patients with severe hepatic disease.